GPCRdb

Ligand source activities (1 row/activity)

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Potency)	# tested GPCRs (Potency)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	44314644	13399	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193573	13399	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL545002	13399	0	None	-	1	Rat	9.1	pEC50	=	9.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314965	12805	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1189070	12805	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL538008	12805	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	533	10	2	5	4.2	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	9937590	107540	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL319460	107540	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL545465	107540	0	None	-	1	Rat	9.0	pEC50	=	9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314574	12804	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1189066	12804	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL538004	12804	0	None	-	1	Rat	8.9	pEC50	=	8.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	547	11	2	5	4.6	CCOC(=O)CCC1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	178024	1940	30	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	5867	1940	30	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	CHEMBL13817	1940	30	None	-1	3	Rat	8.8	pEC50	=	8.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	528	8	2	6	1.8	O=C([C@H](NC(=O)C(N)(C)C)COCc1ccccc1)N1CCC2(CC1)CN(c1c2cccc1)S(=O)(=O)C	10.1016/S0960-894X(97)00421-6
	22867267	13586	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194874	13586	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL553478	13586	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44293557	100619	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL294923	100619	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL540001	100619	0	None	-1	2	Rat	8.0	pEC50	=	8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	447	7	2	3	3.7	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	9890375	97818	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL274599	97818	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL558802	97818	0	None	-1	3	Rat	7.9	pEC50	=	7.9	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	458	5	3	3	3.4	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	10026738	162219	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL417182	162219	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	CHEMBL557206	162219	0	None	-1	2	Rat	7.8	pEC50	=	7.8	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	449	7	2	4	2.9	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CCc3ccccc32)CC1	10.1016/S0960-894X(97)00421-6
	44315065	13380	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193375	13380	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL544769	13380	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	9	2	5	3.8	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](CCCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314651	13493	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194179	13493	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL545704	13493	0	None	-	1	Rat	8.7	pEC50	=	8.7	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867284	12998	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1190399	12998	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL540805	12998	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	505	9	3	4	3.8	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867266	12997	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1190394	12997	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL540800	12997	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	519	10	3	4	4.1	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)CC(CCC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314888	13572	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1194776	13572	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL553290	13572	0	None	-	1	Rat	8.6	pEC50	=	8.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	491	8	3	4	3.4	CC(C)(N)C(=O)N[C@H](CCCc1ccccc1)C(=O)N1CCC2(CC1)C[C@@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314948	13352	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1193173	13352	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL544536	13352	0	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314963	13682	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1195548	13682	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL554852	13682	0	None	-	1	Rat	7.6	pEC50	=	7.6	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	9872740	26260	32	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	567	10	4	7	3.6	C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O	10.1016/S0960-894X(97)00421-6
	CHEMBL13600	26260	32	None	-	1	Rat	8.5	pEC50	=	8.5	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	567	10	4	7	3.6	C[C@@H](O)CNC(C)(C)CC(=O)N[C@@H]1CCc2ccccc2N(Cc2ccc(-c3ccccc3-c3nn[nH]n3)cc2)C1=O	10.1016/S0960-894X(97)00421-6
	44314653	13400	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1193574	13400	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL545003	13400	0	None	-	1	Rat	8.4	pEC50	=	8.4	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	493	8	3	5	2.6	CC(C)(N)C(=O)N[C@H](COCc1ccccc1)C(=O)N1CCC2(CC1)C[C@H](C(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	22867262	13865	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL1196866	13865	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	CHEMBL558422	13865	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	516	7	4	4	3.5	CC(C)(N)C(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)N1CCC2(CC1)C[C@@H](CC(=O)O)c1ccccc12	10.1016/S0960-894X(97)00421-6
	44314767	13588	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194891	13588	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL553507	13588	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44314881	13547	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194592	13547	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL552911	13547	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	521	9	2	6	3.0	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](COCc3ccccc3)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	121879	2204	19	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	5868	2204	19	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	CHEMBL308716	2204	19	None	-1	5	Rat	7.2	pEC50	=	7.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	509	7	3	6	3.6	O=C(CC(N)(C)C)N[C@@H]1CCc2c(N(C1=O)Cc1ccc(cc1)c1ccccc1c1nnn[nH]1)cccc2	10.1016/S0960-894X(97)00421-6
	44314642	13527	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1194442	13527	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL552657	13527	0	None	-	1	Rat	8.2	pEC50	=	8.2	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	544	8	3	5	3.9	CCOC(=O)C[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	44315063	13760	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL1196053	13760	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	CHEMBL555821	13760	0	None	-	1	Rat	8.1	pEC50	=	8.1	Functional	Ability to release growth hormone in a rat pituitary cell assayAbility to release growth hormone in a rat pituitary cell assay	ChEMBL	530	7	3	5	3.5	CCOC(=O)[C@@H]1CC2(CCN(C(=O)[C@@H](Cc3c[nH]c4ccccc34)NC(=O)C(C)(C)N)CC2)c2ccccc21	10.1016/S0960-894X(97)00421-6
	1104	1762	0	None	-	1	Rat	9.1	pIC50	=	9.1	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	1122	2661	0	None	-	1	Rat	10.2	pIC50	None	10.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1123	2662	0	None	-	1	Rat	10.2	pIC50	None	10.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1105	1763	0	None	-	1	Rat	8.0	pIC50	None	8	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	1103	1761	0	None	-	1	Rat	8.2	pIC50	None	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126
	CHEMBL440262	1761	0	None	-	1	Rat	8.2	pIC50	None	8.2	Functional	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	1534126

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Ligands					Receptor			Assay information							Chemical information
Sel. page	Common name	GPCRdb ID	#Vendors	Reference ligand	Fold selectivity (Affinity)	# tested GPCRs (Affinity)	Species	p-value (-log)	Type	Activity Relation	Activity Value	Assay Type	Assay Description	Source	Mol weight	Rot Bonds	H don	H acc	LogP	Smiles	DOI
	148124	205370	82	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
	CHEMBL3545252	205370	82	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
	CHEMBL92	205370	82	None	-	1	Human	9.9	pIC50	=	9.9	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	ChEMBL	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	10.1073/pnas.0610860104
	44387407	141294	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	91928715	141294	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL386366	141294	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3354	116	47	46	-12.4	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	1103	1761	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
	CHEMBL440262	1761	0	None	-	0	Rat	9.1	pIC50	=	9.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
	CHEMBL385308	210601	0	None	-	0	Rat	8.7	pIC50	=	8.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL412221	211230	0	None	-	0	Rat	6.0	pIC50	=	6	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL269263	209038	0	None	-	0	Rat	6.0	pIC50	=	6	Binding	Compound was tested to Inhibit [125I]GRF in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]GRF in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL264522	208879	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	44387431	96074	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	91928702	96074	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL262750	96074	0	None	-	0	Rat	7.9	pIC50	=	7.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3441	119	50	48	-15.1	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	44387406	160696	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	91928713	160696	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL411913	160696	0	None	-	0	Rat	6.9	pIC50	=	6.9	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3136	108	44	42	-11.2	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)CC(=O)CCc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL427794	211636	0	None	-	0	Rat	7.8	pIC50	=	7.8	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL413014	211296	0	None	-	0	Rat	7.8	pIC50	=	7.8	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(C)=O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL414943	211415	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL437461	211973	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	44387434	168420	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	91928693	168420	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL439108	168420	0	None	-	0	Rat	7.7	pIC50	=	7.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3497	123	50	48	-13.5	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL269041	209031	0	None	-	0	Rat	6.7	pIC50	=	6.7	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		None	10.1021/jm00088a023
	CHEMBL428284	211685	0	None	-	0	Rat	6.5	pIC50	=	6.5	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@@H](N)CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL439306	212087	0	None	-	0	Rat	6.4	pIC50	=	6.4	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL427665	211615	0	None	-	0	Rat	7.4	pIC50	=	7.4	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)N)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL262536	208795	0	None	-	0	Rat	7.3	pIC50	=	7.3	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL428135	211670	17	None	-	0	Rat	8.3	pIC50	=	8.3	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	44387430	81483	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	91928698	81483	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL216479	81483	0	None	-	0	Rat	8.2	pIC50	=	8.2	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL	3469	121	50	48	-14.3	CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CCCCCN)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL438545	212027	0	None	-	0	Rat	8.1	pIC50	=	8.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL415373	211438	0	None	-	0	Rat	6.1	pIC50	=	6.1	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL266658	208946	0	None	-	0	Rat	8.0	pIC50	=	8.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL265167	208895	11	None	-	0	Rat	8.0	pIC50	=	8.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1c[nH]cn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1c[nH]cn1)C(=O)N[C@@H](CCC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)[C@@H](C)CC)[C@@H](C)O	10.1021/jm00088a023
	CHEMBL412558	211256	0	None	-	0	Rat	7.0	pIC50	=	7.0	Binding	Compound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenatesCompound was tested to Inhibit [125I]-Growth hormone-releasing factor in rat adenopituitary homogenates	ChEMBL		None	None	None		CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](C)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@H](C(=O)N[C@@H](CC(C)C)C(=O)NCC(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@H](C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CO)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O)[C@@H](C)CC)C(C)C)[C@@H](C)O	10.1021/jm00088a023
	148124	205370	82	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
	CHEMBL3545252	205370	82	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
	CHEMBL92	205370	82	None	-	1	Human	8.0	pIC50	=	8.0	Binding	Displacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cellsDisplacement of [125I]JV1-42 from GHRH receptor expressed in human MX1 cells	Drug Central	807	8	5	14	3.3	CC(=O)O[C@@]12CO[C@@H]1C[C@H](O)[C@@]1(C)C(=O)[C@H](O)C3=C(C)[C@@H](OC(=O)[C@H](O)[C@@H](NC(=O)OC(C)(C)C)c4ccccc4)C[C@@](O)([C@@H](OC(=O)c4ccccc4)[C@@H]12)C3(C)C	None
	9114	2087	0	None	-	0	Human	9.9	pIC50	=	9.9	Binding	Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.Measuring displacement of [<sup>12</sup>5I]JV-1-42 in a radioligand binding assay.	Guide to Pharmacology		None	None	None		None	17261802
	1109	2128	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10542394
	1109	2128	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
	1109	2128	0	None	-	1	Rat	10.1	pKi	=	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1107	2126	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	10542394
	1107	2126	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
	1107	2126	0	None	-	1	Rat	10.3	pKi	=	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1110	2129	0	None	-	1	Rat	10.1	pKi	None	10.1	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1115	2134	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
	1116	2135	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
	1121	2660	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1124	2663	0	None	-	1	Rat	10.2	pKi	None	10.2	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1106	2125	0	None	-	1	Rat	10.3	pKi	None	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1118	2656	0	None	-	1	Rat	10.3	pKi	None	10.3	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
	1108	2127	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1111	2130	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1112	2131	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1113	2132	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1114	2133	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1117	2655	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
	1119	2657	0	None	-	1	Rat	10.4	pKi	None	10.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
	1125	278	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	14755056
	1125	278	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
	1125	278	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431
	1125	278	0	None	-	1	Rat	8.4	pKi	None	8.4	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9892695
	1120	2659	0	None	-	1	Rat	9.9	pKi	None	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	7991622
	1120	2659	0	None	-	1	Rat	9.9	pKi	None	9.9	Binding	UnclassifiedUnclassified	Guide to Pharmacology		None	None	None		None	9145431

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Ligand source activities (1 row/activity)