Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 1001 | 613 | 91 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
| 2144 | 613 | 91 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
| CHEMBL610 | 613 | 91 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
| DB04325 | 613 | 91 | None | -11 | 4 | Mouse | 6.0 | pEC50 | = | 6 | Functional | Guide to Pharmacology | 121 | 2 | 1 | 1 | 1.2 | NCCc1ccccc1 | 16878137 | ||
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |