Ligand source activities (1 row/activity)
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Potency) |
# tested GPCRs (Potency) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 3700 | 3356 | 0 | None | 4 | 2 | Human | 10.1 | pEC50 | = | 10.1 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
| 3697 | 3350 | 0 | None | -2 | 2 | Human | 10.7 | pEC50 | = | 10.7 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
| 3699 | 3353 | 0 | None | -1 | 2 | Human | 10.7 | pEC50 | = | 10.7 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
| 3698 | 3351 | 0 | None | 3 | 2 | Human | 12.5 | pEC50 | = | 12.5 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
| Ligands | Receptor | Assay information | Chemical information | ||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Sel. page | Common name |
GPCRdb ID | #Vendors | Reference ligand |
Fold selectivity (Affinity) |
# tested GPCRs (Affinity) |
Species | p-value (-log) |
Type | Activity Relation |
Activity Value |
Assay Type | Assay Description | Source | Mol weight |
Rot Bonds |
H don | H acc | LogP | Smiles | DOI |
| 3699 | 3353 | 0 | None | - | 1 | Human | 8.7 | pKd | = | 8.7 | Binding | Guide to Pharmacology | None | None | None | None | 21909076 | ||||