GPCR CLASS (FAMILY)

Class A (Rhodopsin)

PDB CODE

SPECIES

Homo sapiens

RESOLUTION

3.2 Å

PREFERRED CHAIN

A

REFERENCE

PUBLICATION DATE

June 26, 2019

3D VIEW

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LIGAND INTERACTIONS

LIGANDS

CHEMBL1615159 - Agonist chembl_ligand pubchem ,

2-[[(3R)-4-(4-Tert-butylphenyl)-3-[[2-(4-methoxyphenyl)sulfanyl-5-[methyl(propan-2-yl)sulfamoyl]benzoyl]amino]butanoyl]amino]acetic acid - PAM pubchem

ENDOGENOUS LIGANDS

noradrenaline, L-NOREPINEPHRINE, (-)-noradrenaline, (-)-adrenaline, Zn2+